(2S,3S)-[2-[3-(Acetoxy)-3,4-dihydro-2-(4-methoxyphenyl)-4-oxo-1,5-benzothiazepin-5(2H)-yl]ethyl]methyl-d3-carbamic Acid 1-Chloroethyl Ester
BR
- Product Code: 82867
CAS:
1246812-21-4
| Molecular Weight: | 510.02 g./mol | Molecular Formula: | C₂₄H₂₄D₃ClN₂O₆S |
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| Density: | Storage Condition: | 2-8°C |
Product Description:
This compound is primarily utilized in the field of medicinal chemistry and pharmaceutical research. It serves as a key intermediate in the synthesis of more complex molecules, particularly those targeting therapeutic areas such as cardiovascular diseases and central nervous system disorders. Its structure, which includes a benzothiazepine core, is often associated with calcium channel blocking activity, making it valuable in the development of drugs that regulate calcium ion flow in cells. Additionally, the presence of deuterium (d3) in the molecule enhances its metabolic stability, which is beneficial for pharmacokinetic studies and drug development. The compound is also used in the preparation of prodrugs, where the 1-chloroethyl ester moiety can be cleaved in vivo to release the active drug, improving bioavailability and targeted delivery.
Sizes / Availability / Pricing:
| Size (g) | Availability | Price | Quantity |
|---|---|---|---|
| 0.050 | 10-20 days | €977.19 |
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(2S,3S)-[2-[3-(Acetoxy)-3,4-dihydro-2-(4-methoxyphenyl)-4-oxo-1,5-benzothiazepin-5(2H)-yl]ethyl]methyl-d3-carbamic Acid 1-Chloroethyl Ester
This compound is primarily utilized in the field of medicinal chemistry and pharmaceutical research. It serves as a key intermediate in the synthesis of more complex molecules, particularly those targeting therapeutic areas such as cardiovascular diseases and central nervous system disorders. Its structure, which includes a benzothiazepine core, is often associated with calcium channel blocking activity, making it valuable in the development of drugs that regulate calcium ion flow in cells. Additionally, the presence of deuterium (d3) in the molecule enhances its metabolic stability, which is beneficial for pharmacokinetic studies and drug development. The compound is also used in the preparation of prodrugs, where the 1-chloroethyl ester moiety can be cleaved in vivo to release the active drug, improving bioavailability and targeted delivery.
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