BMS-986158
≥98%
- Product Code: 57682
CAS:
1800340-40-2
Molecular Weight: | 495.62 g./mol | Molecular Formula: | C₃₀H₃₃N₅O₂ |
---|---|---|---|
EC Number: | MDL Number: | ||
Melting Point: | Boiling Point: | ||
Density: | Storage Condition: | 2-8℃ |
Product Description:
BMS-986158 is primarily investigated for its potential in cancer therapy. It functions as a BET (bromodomain and extra-terminal) inhibitor, targeting proteins involved in the regulation of gene expression. By inhibiting BET proteins, it disrupts the transcription of oncogenes, which are crucial for cancer cell growth and survival. This makes it a promising candidate for treating various cancers, including hematologic malignancies and solid tumors. Clinical trials are ongoing to evaluate its efficacy, safety, and optimal dosing in patients, particularly in combination with other anticancer therapies. Its ability to modulate gene expression also opens possibilities for addressing other diseases influenced by epigenetic dysregulation.
Sizes / Availability / Pricing:
Size (g) | Availability | Price | Quantity |
---|---|---|---|
0.001 | 10-20 days | ฿6,930.00 |
+
-
|
0.005 | 10-20 days | ฿11,133.00 |
+
-
|
BMS-986158
BMS-986158 is primarily investigated for its potential in cancer therapy. It functions as a BET (bromodomain and extra-terminal) inhibitor, targeting proteins involved in the regulation of gene expression. By inhibiting BET proteins, it disrupts the transcription of oncogenes, which are crucial for cancer cell growth and survival. This makes it a promising candidate for treating various cancers, including hematologic malignancies and solid tumors. Clinical trials are ongoing to evaluate its efficacy, safety, and optimal dosing in patients, particularly in combination with other anticancer therapies. Its ability to modulate gene expression also opens possibilities for addressing other diseases influenced by epigenetic dysregulation.
Mechanism | - |
Appearance | - |
Longevity | - |
Strength | - |
Storage | - |
Shelf Life | - |
Allergen(s) | - |
Dosage (Range) | - |
Recommended Dosage | - |
Dosage (Per Day) | - |
Recommended Dosage (Per Day) | - |
Mix Method | - |
Heat Resistance | - |
Stable in pH range | - |
Solubility | - |
Product Types | - |
INCI | - |
Cart
No products
Subtotal:
฿0.00
฿0.00
Total :