2,5-Dioxopyrrolidin-1-yl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl carbonate
98%
- Product Code: 130143
CAS:
1255209-41-6
| Molecular Weight: | 375.18 g./mol | Molecular Formula: | C₁₈H₂₂BNO₇ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD32856201 | |
| Melting Point: | Boiling Point: | 488.3±55.0 °C(Predicted) | |
| Density: | 1.28±0.1 g/cm3(Predicted) | Storage Condition: | -20°C, Sealed, Inert Gas |
Product Description:
Used as a key reagent in Suzuki-Miyaura cross-coupling reactions, enabling the formation of carbon-carbon bonds in pharmaceutical and agrochemical synthesis. Its boronate ester group participates in palladium-catalyzed coupling with aryl halides, making it valuable for constructing biaryl motifs found in active pharmaceutical ingredients. The carbonate linker enhances solubility and stability during conjugation processes, particularly in bioconjugation and prodrug design. Commonly employed in late-stage functionalization of complex molecules due to its compatibility with various functional groups and mild reaction conditions.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 0.100 | 10-20 days | £201.97 |
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| 0.250 | 10-20 days | £302.62 |
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| 1.000 | 10-20 days | £819.64 |
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2,5-Dioxopyrrolidin-1-yl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl carbonate
Used as a key reagent in Suzuki-Miyaura cross-coupling reactions, enabling the formation of carbon-carbon bonds in pharmaceutical and agrochemical synthesis. Its boronate ester group participates in palladium-catalyzed coupling with aryl halides, making it valuable for constructing biaryl motifs found in active pharmaceutical ingredients. The carbonate linker enhances solubility and stability during conjugation processes, particularly in bioconjugation and prodrug design. Commonly employed in late-stage functionalization of complex molecules due to its compatibility with various functional groups and mild reaction conditions.
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