EPZ-719
≥98%
- Product Code: 107237
CAS:
2697176-16-0
| Molecular Weight: | 450.57 g./mol | Molecular Formula: | C₂₂H₃₁FN₄O₃S |
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| Density: | Storage Condition: | 2-8°C, sealed, dry |
Product Description:
EPZ-719 is primarily utilized in the field of cancer research, particularly in the study of epigenetic regulation. It functions as a potent and selective inhibitor of the EZH2 enzyme, which is a key component of the Polycomb Repressive Complex 2 (PRC2). By inhibiting EZH2, EPZ-719 disrupts the methylation of histone H3 on lysine 27 (H3K27me3), a modification associated with gene silencing. This action helps in reactivating tumor suppressor genes that are often silenced in various cancers, making it a valuable tool in understanding and potentially treating malignancies such as lymphoma, leukemia, and certain solid tumors. Researchers use EPZ-719 to explore its therapeutic potential and to study the role of EZH2 in cancer progression and epigenetics.
Sizes / Availability / Pricing:
| Size (g) | Availability | Price | Quantity |
|---|---|---|---|
| 0.005 | 10-20 days | ฿76,500.00 |
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| 0.010 | 10-20 days | ฿130,500.00 |
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EPZ-719
EPZ-719 is primarily utilized in the field of cancer research, particularly in the study of epigenetic regulation. It functions as a potent and selective inhibitor of the EZH2 enzyme, which is a key component of the Polycomb Repressive Complex 2 (PRC2). By inhibiting EZH2, EPZ-719 disrupts the methylation of histone H3 on lysine 27 (H3K27me3), a modification associated with gene silencing. This action helps in reactivating tumor suppressor genes that are often silenced in various cancers, making it a valuable tool in understanding and potentially treating malignancies such as lymphoma, leukemia, and certain solid tumors. Researchers use EPZ-719 to explore its therapeutic potential and to study the role of EZH2 in cancer progression and epigenetics.
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