tert-Butyl (2-((4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)sulfonamido)ethyl)carbamate
95%
- Product Code: 131769
CAS:
1014613-14-9
| Molecular Weight: | 426.34 g./mol | Molecular Formula: | C₁₉H₃₁BN₂O₆S |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD28128481 | |
| Melting Point: | Boiling Point: | ||
| Density: | 1.19±0.1 g/cm3(Predicted) | Storage Condition: | 2-8°C, sealed, dry |
Product Description:
Used primarily as an intermediate in pharmaceutical synthesis, especially in the development of protease inhibitors and other bioactive molecules. Its structure contains both a sulfonamide group and a boronic ester, making it valuable in Suzuki-Miyaura cross-coupling reactions for constructing biaryl systems. The Boc-protected amine allows for selective deprotection and further functionalization in multi-step syntheses. Commonly employed in the preparation of enzyme inhibitors, including those targeting serine proteases, due to the ability of the boron-containing moiety to interact with active site residues. Also utilized in medicinal chemistry for the generation of analogs in structure-activity relationship studies.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 100mg | 10-20 days | ฿2,100.00 |
+
-
|
| 250mg | 10-20 days | ฿3,560.00 |
+
-
|
| 1g | 10-20 days | ฿9,600.00 |
+
-
|
tert-Butyl (2-((4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)sulfonamido)ethyl)carbamate
Used primarily as an intermediate in pharmaceutical synthesis, especially in the development of protease inhibitors and other bioactive molecules. Its structure contains both a sulfonamide group and a boronic ester, making it valuable in Suzuki-Miyaura cross-coupling reactions for constructing biaryl systems. The Boc-protected amine allows for selective deprotection and further functionalization in multi-step syntheses. Commonly employed in the preparation of enzyme inhibitors, including those targeting serine proteases, due to the ability of the boron-containing moiety to interact with active site residues. Also utilized in medicinal chemistry for the generation of analogs in structure-activity relationship studies.
| Mechanism | - |
| Appearance | - |
| Longevity | - |
| Strength | - |
| Storage | - |
| Shelf Life | - |
| Allergen(s) | - |
| Dosage (Range) | - |
| Recommended Dosage | - |
| Dosage (Per Day) | - |
| Recommended Dosage (Per Day) | - |
| Mix Method | - |
| Heat Resistance | - |
| Stable in pH range | - |
| Solubility | - |
| Product Types | - |
| INCI | - |
Purchase History for
Loading purchase history...
Cart
No products
Subtotal:
฿0.00
฿0.00
Total :