1-BOC-5-METHYL-1H-INDOLE-2-BORONIC ACID
95%
- Product Code: 150719
CAS:
475102-14-8
| Molecular Weight: | 275.11 g./mol | Molecular Formula: | C₁₄H₁₈BNO₄ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD04114580 | |
| Melting Point: | Boiling Point: | ||
| Density: | Storage Condition: | 2-8°C, sealed, dry |
Product Description:
Used in Suzuki-Miyaura cross-coupling reactions to synthesize biaryl compounds, particularly in the development of pharmaceutical intermediates. The BOC-protected indole scaffold is valuable in medicinal chemistry for constructing nitrogen-containing heterocycles. Its boronic acid functionality allows for mild, selective coupling with aryl halides, making it useful in the synthesis of complex molecules for drug discovery, especially in the preparation of serotonin receptor modulators and other bioactive indole derivatives. The presence of the methyl group enhances electronic and steric properties, influencing coupling efficiency and selectivity.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 250mg | 10-20 days | ฿4,430.00 |
+
-
|
| 1g | 10-20 days | ฿11,950.00 |
+
-
|
| 5g | 10-20 days | ฿41,780.00 |
+
-
|
1-BOC-5-METHYL-1H-INDOLE-2-BORONIC ACID
Used in Suzuki-Miyaura cross-coupling reactions to synthesize biaryl compounds, particularly in the development of pharmaceutical intermediates. The BOC-protected indole scaffold is valuable in medicinal chemistry for constructing nitrogen-containing heterocycles. Its boronic acid functionality allows for mild, selective coupling with aryl halides, making it useful in the synthesis of complex molecules for drug discovery, especially in the preparation of serotonin receptor modulators and other bioactive indole derivatives. The presence of the methyl group enhances electronic and steric properties, influencing coupling efficiency and selectivity.
| Mechanism | - |
| Appearance | - |
| Longevity | - |
| Strength | - |
| Storage | - |
| Shelf Life | - |
| Allergen(s) | - |
| Dosage (Range) | - |
| Recommended Dosage | - |
| Dosage (Per Day) | - |
| Recommended Dosage (Per Day) | - |
| Mix Method | - |
| Heat Resistance | - |
| Stable in pH range | - |
| Solubility | - |
| Product Types | - |
| INCI | - |
Purchase History for
Loading purchase history...
Cart
No products
Subtotal:
฿0.00
฿0.00
Total :