(4-((2-((tert-Butoxycarbonyl)amino)ethyl)carbamoyl)phenyl)boronic acid
98%
- Product Code: 153592
CAS:
860626-05-7
| Molecular Weight: | 308.1 g./mol | Molecular Formula: | C₁₄H₂₁BN₂O₅ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD09258752 | |
| Melting Point: | Boiling Point: | ||
| Density: | Storage Condition: | 2-8°C, Inert Gas |
Product Description:
Used in the synthesis of targeted protein degraders, particularly in PROTACs (Proteolysis Targeting Chimeras), where it serves as a key intermediate for linking E3 ligase ligands to target protein binders via bioorthogonal conjugation strategies. Its boronic acid group enables stable attachment to biomolecules or solid supports, while the Boc-protected amine allows for controlled deprotection and further functionalization. Commonly applied in medicinal chemistry for developing cancer therapeutics and in bioconjugation for diagnostic probes. Also utilized in Suzuki-Miyaura cross-coupling reactions during the preparation of biaryl-containing drug candidates.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 1.000 | 10-20 days | ฿10,100.00 |
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| 5.000 | 10-20 days | ฿35,320.00 |
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(4-((2-((tert-Butoxycarbonyl)amino)ethyl)carbamoyl)phenyl)boronic acid
Used in the synthesis of targeted protein degraders, particularly in PROTACs (Proteolysis Targeting Chimeras), where it serves as a key intermediate for linking E3 ligase ligands to target protein binders via bioorthogonal conjugation strategies. Its boronic acid group enables stable attachment to biomolecules or solid supports, while the Boc-protected amine allows for controlled deprotection and further functionalization. Commonly applied in medicinal chemistry for developing cancer therapeutics and in bioconjugation for diagnostic probes. Also utilized in Suzuki-Miyaura cross-coupling reactions during the preparation of biaryl-containing drug candidates.
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