CTEP (RO4956371)
10mM in DMSO
- Product Code: 157915
CAS:
871362-31-1
| Molecular Weight: | 391.77 g./mol | Molecular Formula: | C₁₉H₁₃ClF₃N₃O |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD22665726 | |
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| Density: | Storage Condition: | -20°C |
Product Description:
CTEP is a selective and potent negative allosteric modulator of the metabotropic glutamate receptor 5 (mGluR5). It has been primarily investigated for its potential in treating neurological and psychiatric disorders. Due to its ability to cross the blood-brain barrier and provide sustained receptor inhibition, CTEP has been used in preclinical research to study conditions such as Fragile X syndrome, autism spectrum disorders, Parkinson’s disease, and levodopa-induced dyskinesia. It has also shown promise in models of anxiety, depression, and drug addiction, particularly in reducing cocaine-seeking behavior. Its long half-life makes it suitable for chronic dosing studies in animal models, supporting its use as a research tool to explore mGluR5-related pathways and therapeutic interventions.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 1ml | 10-20 days | £201.37 |
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CTEP (RO4956371)
CTEP is a selective and potent negative allosteric modulator of the metabotropic glutamate receptor 5 (mGluR5). It has been primarily investigated for its potential in treating neurological and psychiatric disorders. Due to its ability to cross the blood-brain barrier and provide sustained receptor inhibition, CTEP has been used in preclinical research to study conditions such as Fragile X syndrome, autism spectrum disorders, Parkinson’s disease, and levodopa-induced dyskinesia. It has also shown promise in models of anxiety, depression, and drug addiction, particularly in reducing cocaine-seeking behavior. Its long half-life makes it suitable for chronic dosing studies in animal models, supporting its use as a research tool to explore mGluR5-related pathways and therapeutic interventions.
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