2-(1-(Ethylsulfonyl)-3-(4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1H-Pyrazol-1-Yl)Azetidin-3-Yl)Acetonitrile
95%
- Product Code: 185658
CAS:
1919837-50-5
| Molecular Weight: | 380.27 g./mol | Molecular Formula: | C₁₆H₂₅BN₄O₄S |
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| Density: | Storage Condition: | Room temperature |
Product Description:
Used primarily as a key intermediate in the synthesis of pharmaceutical compounds, especially in the development of kinase inhibitors for targeted cancer therapies. Its structure supports cross-coupling reactions via the boronate ester group, enabling efficient construction of complex drug molecules. Commonly employed in Suzuki-Miyaura coupling reactions during medicinal chemistry research to generate diverse analogs for structure-activity relationship studies. Its nitrile and sulfone functionalities enhance binding selectivity and metabolic stability in final active pharmaceutical ingredients. Widely applied in late-stage functionalization due to its compatibility with various reaction conditions, making it valuable in oncology drug discovery programs.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 1.000 G | 10-20 days | ฿1,700.00 |
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| 5.000 G | 10-20 days | ฿6,610.00 |
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2-(1-(Ethylsulfonyl)-3-(4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1H-Pyrazol-1-Yl)Azetidin-3-Yl)Acetonitrile
Used primarily as a key intermediate in the synthesis of pharmaceutical compounds, especially in the development of kinase inhibitors for targeted cancer therapies. Its structure supports cross-coupling reactions via the boronate ester group, enabling efficient construction of complex drug molecules. Commonly employed in Suzuki-Miyaura coupling reactions during medicinal chemistry research to generate diverse analogs for structure-activity relationship studies. Its nitrile and sulfone functionalities enhance binding selectivity and metabolic stability in final active pharmaceutical ingredients. Widely applied in late-stage functionalization due to its compatibility with various reaction conditions, making it valuable in oncology drug discovery programs.
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