4-Fluoro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole
98%
- Product Code: 188859
CAS:
1256359-96-2
| Molecular Weight: | 261.10 g./mol | Molecular Formula: | C₁₄H₁₇BFNO₂ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD16618972 | |
| Melting Point: | Boiling Point: | ||
| Density: | Storage Condition: | 2-8°C, Inert Gas |
Product Description:
Used primarily as a key intermediate in pharmaceutical synthesis, especially in Suzuki-Miyaura cross-coupling reactions to construct biaryl frameworks. Its indole core with a boronate ester group enables selective carbon-carbon bond formation, making it valuable in the development of bioactive molecules and drug candidates targeting neurological disorders, inflammation, and cancer. The fluorine substituent enhances binding affinity and metabolic stability in final active compounds, improving their pharmacokinetic profile. Commonly employed in research laboratories and early-stage drug discovery for generating novel indole derivatives with tailored biological activities.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 250mg | 10-20 days | ฿4,270.00 |
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| 1g | 10-20 days | ฿11,500.00 |
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| 5g | 10-20 days | ฿40,250.00 |
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| 100mg | 10-20 days | ฿2,630.00 |
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4-Fluoro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole
Used primarily as a key intermediate in pharmaceutical synthesis, especially in Suzuki-Miyaura cross-coupling reactions to construct biaryl frameworks. Its indole core with a boronate ester group enables selective carbon-carbon bond formation, making it valuable in the development of bioactive molecules and drug candidates targeting neurological disorders, inflammation, and cancer. The fluorine substituent enhances binding affinity and metabolic stability in final active compounds, improving their pharmacokinetic profile. Commonly employed in research laboratories and early-stage drug discovery for generating novel indole derivatives with tailored biological activities.
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| Stable in pH range | - |
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