3-(2,6-Difluoro-3,5-dimethoxyphenyl)-1-ethyl-1,3,4,7-tetrahydro-2H-pyrrolo[3',2':5,6]pyrido[4,3-d]pyrimidin-2-one
98%
- Product Code: 192050
CAS:
1513857-72-1
Molecular Weight: | 388.37 g./mol | Molecular Formula: | C₁₉H₁₈F₂N₄O₃ |
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EC Number: | MDL Number: | MFCD33023486 | |
Melting Point: | Boiling Point: | ||
Density: | Storage Condition: | 2-8°C |
Product Description:
Used primarily in pharmaceutical research as a potent and selective inhibitor of phosphodiesterase 10A (PDE10A), this compound is investigated for its potential in treating central nervous system disorders, particularly schizophrenia and other psychiatric conditions involving dysregulated dopamine signaling. By modulating cAMP and cGMP levels in the brain, it helps restore balance in neuronal pathways associated with cognition, motivation, and behavior. Its high blood-brain barrier permeability and favorable metabolic stability make it suitable for in vivo studies aimed at understanding PDE10A's role in neurobiology. It is not used clinically but serves as a valuable tool compound in target validation and proof-of-concept studies for novel antipsychotic therapies.
Sizes / Availability / Pricing:
Size | Availability | Price | Quantity |
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1.000 G | 10-20 days | ฿35,000.00 |
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3-(2,6-Difluoro-3,5-dimethoxyphenyl)-1-ethyl-1,3,4,7-tetrahydro-2H-pyrrolo[3',2':5,6]pyrido[4,3-d]pyrimidin-2-one
Used primarily in pharmaceutical research as a potent and selective inhibitor of phosphodiesterase 10A (PDE10A), this compound is investigated for its potential in treating central nervous system disorders, particularly schizophrenia and other psychiatric conditions involving dysregulated dopamine signaling. By modulating cAMP and cGMP levels in the brain, it helps restore balance in neuronal pathways associated with cognition, motivation, and behavior. Its high blood-brain barrier permeability and favorable metabolic stability make it suitable for in vivo studies aimed at understanding PDE10A's role in neurobiology. It is not used clinically but serves as a valuable tool compound in target validation and proof-of-concept studies for novel antipsychotic therapies.
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