1-Cyclopropyl-6-oxo-1,6-dihydropyridine-3-boronic Acid Pinacol Ester
98%
- Product Code: 192628
CAS:
1596367-55-3
| Molecular Weight: | 261.12 g./mol | Molecular Formula: | C₁₄H₂₀BNO₃ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD16996103 | |
| Melting Point: | Boiling Point: | 326.6±52.0 °C(Predicted) | |
| Density: | 1.13±0.1 g/cm3(Predicted) | Storage Condition: | 2-8°C, Sealed, Inert Gas |
Product Description:
Used as a key intermediate in Suzuki-Miyaura cross-coupling reactions for the synthesis of biologically active compounds, particularly in pharmaceutical development. Its boronic ester group enables efficient carbon-carbon bond formation under mild conditions, making it valuable in constructing complex heterocyclic systems. Commonly employed in the preparation of kinase inhibitors and other drug candidates where the pyridine scaffold is essential for target binding. The cyclopropyl group enhances metabolic stability and influences molecular conformation, contributing to improved potency and selectivity in final active compounds.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 0.050 G | 10-20 days | ฿12,250.00 |
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| 0.100 G | 10-20 days | ฿22,080.00 |
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| 0.250 G | 10-20 days | ฿37,550.00 |
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1-Cyclopropyl-6-oxo-1,6-dihydropyridine-3-boronic Acid Pinacol Ester
Used as a key intermediate in Suzuki-Miyaura cross-coupling reactions for the synthesis of biologically active compounds, particularly in pharmaceutical development. Its boronic ester group enables efficient carbon-carbon bond formation under mild conditions, making it valuable in constructing complex heterocyclic systems. Commonly employed in the preparation of kinase inhibitors and other drug candidates where the pyridine scaffold is essential for target binding. The cyclopropyl group enhances metabolic stability and influences molecular conformation, contributing to improved potency and selectivity in final active compounds.
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