Methyl (S)-3-(bicyclo[1.1.1]pentan-1-yl)-2-((tert-butoxycarbonyl)amino)propanoate
95%
- Product Code: 233197
CAS:
2095488-04-1
| Molecular Weight: | 269.34 g./mol | Molecular Formula: | C₁₄H₂₃NO₄ |
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| EC Number: | MDL Number: | ||
| Melting Point: | Boiling Point: | 363.5±25.0 °C(Predicted) | |
| Density: | 1.151±0.06 g/cm3(Predicted) | Storage Condition: | Room temperature, seal, dry |
Product Description:
Widely used in medicinal chemistry as a key building block for synthesizing bioactive molecules, particularly in the development of pharmaceuticals where structural rigidity and metabolic stability are desired. The bicyclo[1.1.1]pentane (BCP) group acts as a bioisostere for phenyl or tert-butyl groups, improving pharmacokinetic properties such as solubility and resistance to oxidative metabolism. The presence of the Boc-protected amine and methyl ester allows for sequential deprotection and coupling reactions, making it valuable in peptide-like scaffold construction. It is frequently employed in drug discovery programs targeting CNS disorders, oncology, and inflammatory diseases due to its favorable physicochemical properties and ability to modulate target binding affinity.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
|---|---|---|---|
| 50mg | 10-20 days | $1,002.99 |
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| 100mg | 10-20 days | $1,704.76 |
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Methyl (S)-3-(bicyclo[1.1.1]pentan-1-yl)-2-((tert-butoxycarbonyl)amino)propanoate
Widely used in medicinal chemistry as a key building block for synthesizing bioactive molecules, particularly in the development of pharmaceuticals where structural rigidity and metabolic stability are desired. The bicyclo[1.1.1]pentane (BCP) group acts as a bioisostere for phenyl or tert-butyl groups, improving pharmacokinetic properties such as solubility and resistance to oxidative metabolism. The presence of the Boc-protected amine and methyl ester allows for sequential deprotection and coupling reactions, making it valuable in peptide-like scaffold construction. It is frequently employed in drug discovery programs targeting CNS disorders, oncology, and inflammatory diseases due to its favorable physicochemical properties and ability to modulate target binding affinity.
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