Tert-butyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)piperidin-1-carboxylate
97%
- Product Code: 240412
CAS:
1048970-17-7
| Molecular Weight: | 311.23 g./mol | Molecular Formula: | C₁₆H₃₀BNO₄ |
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| EC Number: | MDL Number: | MFCD09997792 | |
| Melting Point: | Boiling Point: | ||
| Density: | Storage Condition: | 2~8℃, dry, sealed |
Product Description:
Widely used in cross-coupling reactions, particularly in Suzuki-Miyaura coupling, to introduce piperidine moieties into complex molecules. This compound serves as a key building block in pharmaceutical synthesis, enabling the construction of nitrogen-containing heterocycles found in bioactive molecules. Its boronate ester group allows for efficient and selective bond formation under mild conditions, making it valuable in drug discovery and development. The tert-butyl carbamate (Boc) protection ensures stability of the piperidine nitrogen during reactions, which can be later deprotected to release the free amine for further functionalization. Commonly employed in the synthesis of central nervous system agents, kinase inhibitors, and other therapeutic targets.
Sizes / Availability / Pricing:
| Size | Availability | Price | Quantity |
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| 5.000 | 10-20 days | $64.31 |
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| 10.000 | 10-20 days | $108.83 |
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| 25.000 | 10-20 days | $242.39 |
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| 100.000 | 10-20 days | $905.25 |
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| 50.000 | 10-20 days | $468.70 |
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Tert-butyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)piperidin-1-carboxylate
Widely used in cross-coupling reactions, particularly in Suzuki-Miyaura coupling, to introduce piperidine moieties into complex molecules. This compound serves as a key building block in pharmaceutical synthesis, enabling the construction of nitrogen-containing heterocycles found in bioactive molecules. Its boronate ester group allows for efficient and selective bond formation under mild conditions, making it valuable in drug discovery and development. The tert-butyl carbamate (Boc) protection ensures stability of the piperidine nitrogen during reactions, which can be later deprotected to release the free amine for further functionalization. Commonly employed in the synthesis of central nervous system agents, kinase inhibitors, and other therapeutic targets.
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