Pinacol 6-bromo-1-boc-indole-3-borate
95%
- Product Code: 49822
CAS:
1218790-27-2
| Molecular Weight: | 422.12 g./mol | Molecular Formula: | C₁₉H₂₅BBrNO₄ |
|---|---|---|---|
| EC Number: | MDL Number: | MFCD15143608 | |
| Melting Point: | Boiling Point: | ||
| Density: | Storage Condition: | 2-8℃, dry, airtight |
Product Description:
Pinacol 6-bromo-1-boc-indole-3-borate is primarily utilized in organic synthesis as a key intermediate for constructing complex indole derivatives. Its borate ester functionality makes it a valuable reagent in cross-coupling reactions, particularly Suzuki-Miyaura couplings, which are widely employed in the synthesis of pharmaceuticals, agrochemicals, and advanced materials. The Boc-protected amine group enhances its stability during reactions, allowing for selective deprotection and further functionalization. Additionally, the bromo substituent at the 6-position provides a reactive site for further modifications, enabling the introduction of diverse substituents to tailor the properties of the final product. This compound is particularly useful in medicinal chemistry for the development of biologically active indole-based compounds, such as kinase inhibitors and serotonin receptor modulators.
Sizes / Availability / Pricing:
| Size (g) | Availability | Price | Quantity |
|---|---|---|---|
| 0.100 | 10-20 days | ฿8,991.00 |
+
-
|
| 0.250 | 10-20 days | ฿14,994.00 |
+
-
|
| 1.000 | 10-20 days | ฿39,924.00 |
+
-
|
Pinacol 6-bromo-1-boc-indole-3-borate
Pinacol 6-bromo-1-boc-indole-3-borate is primarily utilized in organic synthesis as a key intermediate for constructing complex indole derivatives. Its borate ester functionality makes it a valuable reagent in cross-coupling reactions, particularly Suzuki-Miyaura couplings, which are widely employed in the synthesis of pharmaceuticals, agrochemicals, and advanced materials. The Boc-protected amine group enhances its stability during reactions, allowing for selective deprotection and further functionalization. Additionally, the bromo substituent at the 6-position provides a reactive site for further modifications, enabling the introduction of diverse substituents to tailor the properties of the final product. This compound is particularly useful in medicinal chemistry for the development of biologically active indole-based compounds, such as kinase inhibitors and serotonin receptor modulators.
| Mechanism | - |
| Appearance | - |
| Longevity | - |
| Strength | - |
| Storage | - |
| Shelf Life | - |
| Allergen(s) | - |
| Dosage (Range) | - |
| Recommended Dosage | - |
| Dosage (Per Day) | - |
| Recommended Dosage (Per Day) | - |
| Mix Method | - |
| Heat Resistance | - |
| Stable in pH range | - |
| Solubility | - |
| Product Types | - |
| INCI | - |
Cart
No products
Subtotal:
฿0.00
฿0.00
Total :