Arteanoflavone exhibits significant biological activity, making it valuable in pharmaceutical and nutraceutical applications. It is studied for its anti-inflammatory and antioxidant properties, which may support its use in managing oxidative stress-related conditions such as neurodegenerative diseases and cardiovascular disorders. Research also indicates potential anticancer effects, where it may inhibit the proliferation of certain tumor cells by inducing apoptosis and suppressing key signaling pathways involved in cancer progression. Due to its natural origin and bioactive profile, arteanoflavone is explored as a lead compound in drug development and as an active ingredient in herbal formulations targeting metabolic and age-related diseases. Additionally, its presence in traditional medicinal plants supports its role in ethnopharmacology, contributing to the validation of plant-based therapies.