Atherosperminine exhibits significant biological activity, making it of interest in pharmaceutical and medicinal research. It has demonstrated potential as an antimicrobial agent, showing inhibitory effects against certain bacterial and fungal strains. Studies also suggest it may possess anti-inflammatory and neuroprotective properties, which could be relevant in developing treatments for neurodegenerative conditions. Additionally, its role in modulating cellular pathways has prompted investigation into its use as a lead compound for drug development. Due to its natural origin and structural complexity, it is also used as a reference substance in phytochemical studies and natural product isolation.