(R)-Azetidin-2-ylmethanol is primarily used in the synthesis of pharmaceutical compounds, particularly in the development of beta-lactam antibiotics. Its structure serves as a key intermediate in creating molecules that exhibit antibacterial properties. Additionally, it is utilized in the preparation of chiral building blocks for drug discovery, enabling the production of enantiomerically pure substances. This compound is also explored in the field of medicinal chemistry for designing inhibitors targeting specific enzymes or receptors, contributing to the development of novel therapeutic agents. Its applications extend to organic synthesis, where it acts as a versatile reagent for constructing complex molecular architectures.