Used in pharmaceutical research as a cyclic dipeptide scaffold for developing bioactive compounds. Shows potential in enhancing metabolic stability and membrane permeability of peptide-based drugs. Investigated for its role in modulating cellular signaling pathways due to its structural rigidity and ability to mimic secondary structures of proteins. Also explored in the design of enzyme inhibitors and receptor ligands. Exhibits antimicrobial and antitumor activities in preliminary studies, making it a candidate for drug discovery. Employed in peptidomimetic chemistry to improve pharmacokinetic properties of therapeutic peptides.