Benzyl 5-oxo-2-azabicyclo[2.2.1]heptane-2-carboxylate is primarily utilized in organic synthesis as a key intermediate in the production of complex molecules. Its bicyclic structure makes it valuable for constructing pharmacologically active compounds, particularly in the development of drugs targeting neurological disorders. The compound is often employed in the synthesis of peptide mimetics, which are crucial for creating enzyme inhibitors and receptor modulators. Additionally, its ester group allows for further functionalization, making it a versatile building block in medicinal chemistry. Researchers also use it in the preparation of chiral catalysts, which are essential for asymmetric synthesis in the pharmaceutical industry.