Alpinumisoflavone exhibits significant biological activities, making it valuable in pharmaceutical and medicinal research. It is studied for its anti-cancer properties, particularly in inhibiting the growth of various tumor cells, including breast and colon cancer, by inducing apoptosis and blocking cell cycle progression. The compound also shows anti-inflammatory effects by suppressing key inflammatory mediators like nitric oxide and prostaglandins, and inhibiting enzymes involved in chronic inflammation. Additionally, alpinumisoflavone demonstrates antimicrobial activity against certain bacteria and fungi, suggesting potential use in treating infections. Its antioxidant properties contribute to cellular protection against oxidative stress, which is relevant in aging and neurodegenerative diseases. Furthermore, it is investigated for its phytoestrogenic effects in modulating hormone balance and supporting bone health, particularly in osteoporosis. Research is ongoing to explore its use in drug development and as a lead compound for synthesizing more potent derivatives.