Valerosidate is primarily used in pharmaceutical research and development due to its potential bioactive properties. It serves as a key intermediate in the synthesis of natural product derivatives with possible sedative and anxiolytic effects. Its structural characteristics make it valuable in studying glycoside-based compounds that influence central nervous system activity. Additionally, valerosidate is investigated for its role in enhancing the stability and solubility of active pharmaceutical ingredients, particularly in formulations targeting neurological disorders. It is also utilized in analytical studies to understand metabolic pathways of related glycosides in plant and animal models.