Stepharine is a bioactive aporphine alkaloid primarily utilized in pharmacology due to its diverse therapeutic properties. It has been studied for its antihypertensive effects, helping to lower blood pressure and supporting the development of treatments for cardiovascular diseases. Additionally, stepharine exhibits anti-inflammatory and analgesic properties, making it a candidate for managing pain, swelling, and chronic inflammatory conditions. Research also explores its interactions with the central nervous system, including modulation of neurotransmitter activity and specific brain receptors, for potential applications in treating neurological disorders such as anxiety and depression. Its historical role in traditional medicine has further sparked interest in broader uses, including possible anticancer activities.