Lobetyolinin is primarily used in traditional medicine and modern herbal formulations due to its bioactive properties. It exhibits anti-inflammatory and antioxidant activities, making it valuable in treating respiratory conditions such as bronchitis and cough. The compound supports immune function and is often included in remedies aimed at improving lung health. It also shows potential in regulating gastrointestinal motility, which helps in managing digestive disorders. Due to its natural origin and low toxicity, it is increasingly studied for use in nutraceuticals and functional health products. Research is ongoing into its neuroprotective effects, particularly in age-related cognitive decline.