Used in pharmaceutical research as a potent and selective antagonist of the GPR135 receptor, which is involved in regulating immune responses and metabolic functions. Shows potential in the development of treatments for inflammatory diseases and certain types of cancer due to its ability to modulate signaling pathways linked to cell proliferation and immune cell activity. Also employed as a biochemical tool to study receptor function in vitro and in animal models. Its structural properties make it suitable for blood-brain barrier penetration, enabling exploration in central nervous system disorders.