Ophiopogonanone C is a homoisoflavonoid compound isolated from Ophiopogon japonicus, used in skincare formulations for its potent antioxidant properties, which help protect skin cells from oxidative stress and environmental damage. It shows significant potential in anti-aging products by supporting cellular health and reducing signs of aging. In herbal and traditional medicine, it is investigated for anti-inflammatory and neuroprotective effects. Additionally, research explores its antiviral activity and possible applications in pharmaceutical development for chronic diseases such as diabetes and neurological disorders. Studies also indicate anti-cancer potential, with in vitro evidence of inhibiting abnormal cell growth in certain cancer cell lines, making it a promising bioactive compound for future therapeutic uses.