Pyrrolo[1,2-b][1,2,5]benzothiadiazepine-8-carboxamide, N-[2-(2R)-1,4-dioxan-2-ylethyl]-10,11-dihydro-2-methyl-11-oxo-, 5,5-dioxide

95%

Reagent Code: #226830
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CAS Number 2243162-67-4

science Other reagents with same CAS 2243162-67-4

blur_circular Chemical Specifications

scatter_plot Molecular Information
Weight 419.5 g/mol
Formula C₁₉H₂₁N₃O₆S
inventory_2 Storage & Handling
Storage 2-8°C, dry, closed

description Product Description

Used in pharmaceutical research as a potent and selective antagonist of the GABA-A receptor, particularly targeting α5 subunit-containing receptors. This compound is investigated for its potential to enhance cognitive function and memory, especially in conditions like Alzheimer’s disease and other cognitive impairments. Due to its ability to modulate inhibitory neurotransmission without inducing anxiety or seizures—common side effects with non-selective GABA-A antagonists—it serves as a valuable tool in neuroscience for studying synaptic plasticity and neural circuits. Its structural properties also make it a lead candidate in developing nootropic drugs with improved safety profiles.

Available Sizes & Pricing

Size Availability Unit Price Quantity
5mg
10-20 days ฿86,940.00
Pyrrolo[1,2-b][1,2,5]benzothiadiazepine-8-carboxamide, N-[2-(2R)-1,4-dioxan-2-ylethyl]-10,11-dihydro-2-methyl-11-oxo-, 5,5-dioxide
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Used in pharmaceutical research as a potent and selective antagonist of the GABA-A receptor, particularly targeting α5 subunit-containing receptors. This compound is investigated for its potential to enhance cognitive function and memory, especially in conditions like Alzheimer’s disease and other cognitive impairments. Due to its ability to modulate inhibitory neurotransmission without inducing anxiety or seizures—common side effects with non-selective GABA-A antagonists—it serves as a valuable tool in

Used in pharmaceutical research as a potent and selective antagonist of the GABA-A receptor, particularly targeting α5 subunit-containing receptors. This compound is investigated for its potential to enhance cognitive function and memory, especially in conditions like Alzheimer’s disease and other cognitive impairments. Due to its ability to modulate inhibitory neurotransmission without inducing anxiety or seizures—common side effects with non-selective GABA-A antagonists—it serves as a valuable tool in neuroscience for studying synaptic plasticity and neural circuits. Its structural properties also make it a lead candidate in developing nootropic drugs with improved safety profiles.

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