Gigantol is a naturally occurring compound with various applications in the fields of medicine and pharmacology. It has been studied for its potential anti-cancer properties, showing promise in inhibiting the growth of certain cancer cells by inducing apoptosis and suppressing tumor progression. Additionally, gigantol exhibits anti-inflammatory and antioxidant effects, making it a candidate for treating inflammatory diseases and reducing oxidative stress-related damage in cells. In traditional medicine, it has been used for its analgesic properties to alleviate pain. Research also suggests its potential in combating microbial infections, including those caused by drug-resistant bacteria, due to its antimicrobial activity. Furthermore, gigantol has been explored for its neuroprotective effects, potentially aiding in the treatment of neurodegenerative disorders like Alzheimer’s disease. Preliminary studies also indicate its anti-diabetic potential, which may help in managing diabetes through mechanisms such as improving insulin sensitivity. Its diverse biological activities make it a compound of interest for developing new therapeutic agents.